AG 99
CAS No. 122520-85-8
AG 99 ( (E)-Tyrphostin AG 99;(E)-Tyrphostin 46;Tyrphostin 46 )
Catalog No. M19940 CAS No. 122520-85-8
AG-99 is an inhibitor of EGFR kinase (IC50: 10 μM in the human epidermoid carcinoma cell line A431).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
5MG | 27 | In Stock |
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10MG | 42 | In Stock |
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25MG | 66 | In Stock |
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50MG | 87 | In Stock |
|
100MG | 147 | In Stock |
|
200MG | Get Quote | In Stock |
|
500MG | Get Quote | In Stock |
|
1G | Get Quote | In Stock |
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Biological Information
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Product NameAG 99
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NoteResearch use only not for human use.
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Brief DescriptionAG-99 is an inhibitor of EGFR kinase (IC50: 10 μM in the human epidermoid carcinoma cell line A431).
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DescriptionAG-99 is an inhibitor of EGFR kinase (IC50: 10 μM in the human epidermoid carcinoma cell line A431).
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Synonyms(E)-Tyrphostin AG 99;(E)-Tyrphostin 46;Tyrphostin 46
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PathwayAngiogenesis
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TargetEGFR
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RecptorEGFR
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Research Area——
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Indication——
Chemical Information
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CAS Number122520-85-8
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Formula Weight204.18
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Molecular FormulaC10H8N2O3
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Purity>98% (HPLC)
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SolubilityDMSO: 20 mg/mL;Ethanol: 1 mg/mL;Water: Insoluble
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SMILESNC(=O)C(=C\c1ccc(O)c(O)c1)\C#N
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Gazit A et al. Tyrphostins. 6. Dimeric benzylidenemalononitrile tyrophostins: potent inhibitors of EGF receptor tyrosine kinase in vitro. J Med Chem. 1996 Dec 6;39(25):4905-11.
molnova catalog
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